Sfoglia per Autore
MIBE acts as antagonist ligand of both estrogen receptor alpha and GPER in breast cancer cells
2012-01-01 Lappano, R.; Santolla, M. F.; Pupo, M.; Sinicropi, M. S.; Caruso, A.; Rosano, C.; Maggiolini, M.
Two Novel GPER Agonists Induce Gene Expression Changes and Growth Effects in Cancer Cells.
2012-01-01 Lappano, R; Rosano, C; Santolla, Mf; Pupo, M; De Francesco, Em; De Marco, P; Ponassi, M; Spallarossa, A; Ranise, A; Maggiolini, Marcello
Recent Advances in the Rationale Design of GPER Ligands.
2012-01-01 Rosano, C; Lappano, R; Santolla, Mf; Ponassi, M; Donadini, A; Maggiolini, Marcello
Bisphenol A Induces Gene Expression Changes and Proliferative Effects through GPER in Breast Cancer Cells and Cancer-Associated Fibroblasts
2012-01-01 Pupo, M; Pisano, A; Lappano, R; Santolla, Mf; De Francesco, Em; Abonante, S; Rosano, C; Maggiolini, Marcello
G protein-coupled estrogen receptor mediates the up-regulation of fatty acid synthase induced by 17β-estradiol in cancer cells and cancer-associated fibroblasts
2012-01-01 Santolla, Mf; Lappano, R; De Marco, P; Pupo, M; Vivacqua, A; Sisci, D; Abonante, S; Iacopetta, D; Cappello, Ar; Dolce, V; Maggiolini, M
Carbazole derivatives as potential novel agonist of GPER
2013-01-01 Sinicropi, Maria Stefania; Lappano, R; Caruso, A; Santolla, M. F.; Pisano, A; Rosano, C; Capasso, A; Panno, A; Lancelot, J. C.; Rault, S; Saturnino, C; Maggiolini, M; Angelamaria Caporale, A.
Nuovi ligandi di recettori estrogenici accoppiati a proteina G
2013-01-01 Maggiolini, Marcello; Santolla, Mf
Insulin-like growth factor-I regulates GPER expression and function in cancer cells
2013-01-01 De Marco, P; Bartella, V; Vivacqua, Adele; Lappano, R; Santolla, Mf; Morcavallo, A; Pezzi, Vincenzo; Belfiore, A; Maggiolini, Marcello
HIF-1α/GPER signaling mediates the expression of VEGF induced by hypoxia in breast cancer associated fibroblasts (CAFs)
2013-01-01 De Francesco, Em; Lappano, R; Santolla, Mf; Marsico, Stefania; Caruso, A; Maggiolini, Marcello
Oleuropeina ed idrossitirisolo attivano pathways GPER-dipendenti inducendo apoptosi in cellule tumorali mammarie SKBR3 negative per i recettori estrogenici α e β.
2013-01-01 Chimento, Adele; Casaburi, Ivan; Rosano, Camillo; Avena, Paola; DE LUCA, Arianna; Campana, Carmela; Martire, Emilia; Santolla, Maria Francesca; Maggiolini, Marcello; Pezzi, Vincenzo; Sirianni, Rosa.
Identification of two novel benzo[b]pyrrolo[1,2-d][1,4]oxazin-4-one derivatives acting as GPER antagonists
2014-01-01 Grande, Fedora; Avino, S; Santolla, Mf; Aiello, A; Perri, Mg; Rosano, C; Badolato, M; Vigliatore, F; Garofalo, A; Maggiolini, M.
GPER mediates activation of HIF1α/VEGF signaling by estrogens
2014-01-01 DE FRANCESCO, Ernestina Marianna; Pellegrino, M; Santolla, Mf; Lappano, R; Ricchio, E; Abonante, S; Maggiolini, Marcello
Niacin activates the G protein estrogen receptor (GPER)-mediated signalling
2014-01-01 Santolla, Maria Francesca; De Francesco, Em; Lappano, R; Rosano, C; Abonante, S; Maggiolini, Marcello
Oleuropein and hydroxytyrosol activate GPER/ GPR30-dependent pathways leading to apoptosis of ER-negative SKBR3 breast cancer cells
2014-01-01 Chimento, Adele; Casaburi, Ivan; Rosano, C; Avena, P; De Luca, A; Campana, C; Martire, E; Santolla, Mf; Maggiolini, Marcello; Pezzi, Vincenzo; Sirianni, Rosa
A calixpyrrole derivative acts as an antagonist to GPER, a G-protein coupled receptor: mechanisms and models.
2015-01-01 Lappano, R; Rosano, C; Pisano, A; Santolla, Mf; De Francesco, Em; De Marco, P; Dolce, Vincenza; Ponassi, M; Felli, L; Cafeo, G; Kohnke, Fh; Abonante, S; Maggiolini, Marcello
Copper activates HIF-1α/GPER/VEGF signalling in cancer cells
2015-01-01 Rigiracciolo, Dc; Scarpelli, A; Lappano, R; Pisano, A; Santolla, MARIA FRANCESCA; De Marco, P; Cirillo, F; Cappello, Anna Rita; Dolce, Vincenza; Belfiore, A; Maggiolini, Marcello; De Francesco, Em
(6-Bromo-1,4-dimethyl-9H-carbazol-3-yl-methylene)-hydrazine (Carbhydraz) Acts as a GPER Agonist in Breast Cancer Cells
2015-01-01 Sinicropi, M. S.; Lappano, R.; Caruso, A.; Santolla, M. F.; Pisano, A.; Rosano, C.; Capasso, A.; Panno, A.; Lancelot, J. C.; Rault, S.; Saturnino, C.; Maggiolini, M.
A Bodipy as a luminescent probe for detection of the G protein estrogen receptor (GPER)
2015-01-01 Papalia, T; Lappano, R; Barattucci, A; Pisano, A; Bruno, G; Santolla, Mf; Campagna, S; De Marco, P; Puntoriero, F; De Francesco, Em; Rosano, C; Maggiolini, Marcello; Bonaccorsi, P.
SIRT1 is involved in oncogenic signaling mediated by GPER in breast cancer
2015-01-01 Santolla, Mf; Avino, S; Pellegrino, M; De Francesco, Em; De Marco, P; Lappano, R; Vivacqua, Adele; Cirillo, F; Rigiracciolo, Dc; Scarpelli, A; Abonante, S; Maggiolini, Marcello
Identification of two benzopyrroloxazines acting as selective GPER antagonists in breast cancer cells and cancer-associated fibroblasts
2015-01-01 Maggiolini, Marcello; Santolla, Mf; Avino, S; Aiello, Francesca; Rosano, C; Garofalo, Antonio; Grande, Fedora
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
MIBE acts as antagonist ligand of both estrogen receptor alpha and GPER in breast cancer cells | 1-gen-2012 | Lappano, R.; Santolla, M. F.; Pupo, M.; Sinicropi, M. S.; Caruso, A.; Rosano, C.; Maggiolini, M. | |
Two Novel GPER Agonists Induce Gene Expression Changes and Growth Effects in Cancer Cells. | 1-gen-2012 | Lappano, R; Rosano, C; Santolla, Mf; Pupo, M; De Francesco, Em; De Marco, P; Ponassi, M; Spallarossa, A; Ranise, A; Maggiolini, Marcello | |
Recent Advances in the Rationale Design of GPER Ligands. | 1-gen-2012 | Rosano, C; Lappano, R; Santolla, Mf; Ponassi, M; Donadini, A; Maggiolini, Marcello | |
Bisphenol A Induces Gene Expression Changes and Proliferative Effects through GPER in Breast Cancer Cells and Cancer-Associated Fibroblasts | 1-gen-2012 | Pupo, M; Pisano, A; Lappano, R; Santolla, Mf; De Francesco, Em; Abonante, S; Rosano, C; Maggiolini, Marcello | |
G protein-coupled estrogen receptor mediates the up-regulation of fatty acid synthase induced by 17β-estradiol in cancer cells and cancer-associated fibroblasts | 1-gen-2012 | Santolla, Mf; Lappano, R; De Marco, P; Pupo, M; Vivacqua, A; Sisci, D; Abonante, S; Iacopetta, D; Cappello, Ar; Dolce, V; Maggiolini, M | |
Carbazole derivatives as potential novel agonist of GPER | 1-gen-2013 | Sinicropi, Maria Stefania; Lappano, R; Caruso, A; Santolla, M. F.; Pisano, A; Rosano, C; Capasso, A; Panno, A; Lancelot, J. C.; Rault, S; Saturnino, C; Maggiolini, M; Angelamaria Caporale, A. | |
Nuovi ligandi di recettori estrogenici accoppiati a proteina G | 1-gen-2013 | Maggiolini, Marcello; Santolla, Mf | |
Insulin-like growth factor-I regulates GPER expression and function in cancer cells | 1-gen-2013 | De Marco, P; Bartella, V; Vivacqua, Adele; Lappano, R; Santolla, Mf; Morcavallo, A; Pezzi, Vincenzo; Belfiore, A; Maggiolini, Marcello | |
HIF-1α/GPER signaling mediates the expression of VEGF induced by hypoxia in breast cancer associated fibroblasts (CAFs) | 1-gen-2013 | De Francesco, Em; Lappano, R; Santolla, Mf; Marsico, Stefania; Caruso, A; Maggiolini, Marcello | |
Oleuropeina ed idrossitirisolo attivano pathways GPER-dipendenti inducendo apoptosi in cellule tumorali mammarie SKBR3 negative per i recettori estrogenici α e β. | 1-gen-2013 | Chimento, Adele; Casaburi, Ivan; Rosano, Camillo; Avena, Paola; DE LUCA, Arianna; Campana, Carmela; Martire, Emilia; Santolla, Maria Francesca; Maggiolini, Marcello; Pezzi, Vincenzo; Sirianni, Rosa. | |
Identification of two novel benzo[b]pyrrolo[1,2-d][1,4]oxazin-4-one derivatives acting as GPER antagonists | 1-gen-2014 | Grande, Fedora; Avino, S; Santolla, Mf; Aiello, A; Perri, Mg; Rosano, C; Badolato, M; Vigliatore, F; Garofalo, A; Maggiolini, M. | |
GPER mediates activation of HIF1α/VEGF signaling by estrogens | 1-gen-2014 | DE FRANCESCO, Ernestina Marianna; Pellegrino, M; Santolla, Mf; Lappano, R; Ricchio, E; Abonante, S; Maggiolini, Marcello | |
Niacin activates the G protein estrogen receptor (GPER)-mediated signalling | 1-gen-2014 | Santolla, Maria Francesca; De Francesco, Em; Lappano, R; Rosano, C; Abonante, S; Maggiolini, Marcello | |
Oleuropein and hydroxytyrosol activate GPER/ GPR30-dependent pathways leading to apoptosis of ER-negative SKBR3 breast cancer cells | 1-gen-2014 | Chimento, Adele; Casaburi, Ivan; Rosano, C; Avena, P; De Luca, A; Campana, C; Martire, E; Santolla, Mf; Maggiolini, Marcello; Pezzi, Vincenzo; Sirianni, Rosa | |
A calixpyrrole derivative acts as an antagonist to GPER, a G-protein coupled receptor: mechanisms and models. | 1-gen-2015 | Lappano, R; Rosano, C; Pisano, A; Santolla, Mf; De Francesco, Em; De Marco, P; Dolce, Vincenza; Ponassi, M; Felli, L; Cafeo, G; Kohnke, Fh; Abonante, S; Maggiolini, Marcello | |
Copper activates HIF-1α/GPER/VEGF signalling in cancer cells | 1-gen-2015 | Rigiracciolo, Dc; Scarpelli, A; Lappano, R; Pisano, A; Santolla, MARIA FRANCESCA; De Marco, P; Cirillo, F; Cappello, Anna Rita; Dolce, Vincenza; Belfiore, A; Maggiolini, Marcello; De Francesco, Em | |
(6-Bromo-1,4-dimethyl-9H-carbazol-3-yl-methylene)-hydrazine (Carbhydraz) Acts as a GPER Agonist in Breast Cancer Cells | 1-gen-2015 | Sinicropi, M. S.; Lappano, R.; Caruso, A.; Santolla, M. F.; Pisano, A.; Rosano, C.; Capasso, A.; Panno, A.; Lancelot, J. C.; Rault, S.; Saturnino, C.; Maggiolini, M. | |
A Bodipy as a luminescent probe for detection of the G protein estrogen receptor (GPER) | 1-gen-2015 | Papalia, T; Lappano, R; Barattucci, A; Pisano, A; Bruno, G; Santolla, Mf; Campagna, S; De Marco, P; Puntoriero, F; De Francesco, Em; Rosano, C; Maggiolini, Marcello; Bonaccorsi, P. | |
SIRT1 is involved in oncogenic signaling mediated by GPER in breast cancer | 1-gen-2015 | Santolla, Mf; Avino, S; Pellegrino, M; De Francesco, Em; De Marco, P; Lappano, R; Vivacqua, Adele; Cirillo, F; Rigiracciolo, Dc; Scarpelli, A; Abonante, S; Maggiolini, Marcello | |
Identification of two benzopyrroloxazines acting as selective GPER antagonists in breast cancer cells and cancer-associated fibroblasts | 1-gen-2015 | Maggiolini, Marcello; Santolla, Mf; Avino, S; Aiello, Francesca; Rosano, C; Garofalo, Antonio; Grande, Fedora |
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