Sfoglia per Autore
Toward multitasking pharmacological COX-targeting agents: Non-steroidal anti-inflammatory prodrugs with antiproliferative effects
2021-01-01 Grande, F.; Giordano, F.; Occhiuzzi, M. A.; Rocca, C.; Ioele, G.; De Luca, M.; Ragno, G.; Panno, M. L.; Rizzuti, B.; Garofalo, A.
Sub-micromolar inhibition of sars-cov-2 3clpro by natural compounds
2021-01-01 Rizzuti, B.; Ceballos-Laita, L.; Ortega-Alarcon, D.; Jimenez-Alesanco, A.; Vega, S.; Grande, F.; Conforti, F.; Abian, O.; Velazquez-Campoy, A.
Polyphenols from citrus tacle® extract endowed with hmgcr inhibitory activity: An antihypercholesterolemia natural remedy
2021-01-01 Grande, F.; Occhiuzzi, M. A.; Perri, M. R.; Ioele, G.; Rizzuti, B.; Statti, G.; Garofalo, A.
A single evolutionarily divergent mutation determines the different FAD-binding affinities of human and rat NQO1 due to site-specific phosphorylation
2022-01-01 Pacheco-Garcia, J. L.; Loginov, D.; Rizzuti, B.; Vankova, P.; Neira, J. L.; Kavan, D.; Mesa-Torres, N.; Guzzi, R.; Man, P.; Pey, A. L.
Interaction of letrozole and its degradation products with aromatase: chemometric assessment of kinetics and structure-based binding validation
2022-01-01 De Luca, Michele; Occhiuzzi, Maria Antonietta; Rizzuti, Bruno; Ioele, Giuseppina; Ragno, Gaetano; Garofalo, Antonio; Grande, Fedora
The interaction of tryptophan enantiomers with model membranes is modulated by polar head type and physical state of phospholipids
2023-01-01 Guglielmelli, Alexa; Bartucci, Rosa; Rizzuti, Bruno; Palermo, Giovanna; Guzzi, Rita; Strangi, Giuseppe
Promising Perspectives of the Antiproliferative GPER Inverse Agonist ERα17p in Breast Cancer
2023-01-01 Kampa, Marilena; Lappano, Rosamaria; Grande, Fedora; Rizzuti, Bruno; Maggiolini, Marcello; Castanas, Elias; Jacquot, Yves
Targeting of mitochondrial fission through natural flavanones elicits anti-myeloma activity
2024-01-01 Torcasio, Roberta; Gallo Cantafio, Maria Eugenia; Veneziano, Claudia; De Marco, Carmela; Ganino, Ludovica; Valentino, Ilenia; Occhiuzzi, Maria Antonietta; Perrotta, Ida Daniela; Mancuso, Teresa; Conforti, Filomena; Rizzuti, Bruno; Martino, Enrica Antonia; Gentile, Massimo; Neri, Antonino; Viglietto, Giuseppe; Grande, Fedora; Amodio, Nicola
Dissecting CYP1A2 Activation by Arylalkanoic Acid Prodrugs toward the Development of Anti-Inflammatory Agents
2024-01-01 Occhiuzzi, Maria Antonietta; Ioele, Giuseppina; De Luca, Michele; Rizzuti, Bruno; Scordamaglia, Domenica; Lappano, Rosamaria; Maggiolini, Marcello; Garofalo, Antonio; Grande, Fedora
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Toward multitasking pharmacological COX-targeting agents: Non-steroidal anti-inflammatory prodrugs with antiproliferative effects | 1-gen-2021 | Grande, F.; Giordano, F.; Occhiuzzi, M. A.; Rocca, C.; Ioele, G.; De Luca, M.; Ragno, G.; Panno, M. L.; Rizzuti, B.; Garofalo, A. | |
Sub-micromolar inhibition of sars-cov-2 3clpro by natural compounds | 1-gen-2021 | Rizzuti, B.; Ceballos-Laita, L.; Ortega-Alarcon, D.; Jimenez-Alesanco, A.; Vega, S.; Grande, F.; Conforti, F.; Abian, O.; Velazquez-Campoy, A. | |
Polyphenols from citrus tacle® extract endowed with hmgcr inhibitory activity: An antihypercholesterolemia natural remedy | 1-gen-2021 | Grande, F.; Occhiuzzi, M. A.; Perri, M. R.; Ioele, G.; Rizzuti, B.; Statti, G.; Garofalo, A. | |
A single evolutionarily divergent mutation determines the different FAD-binding affinities of human and rat NQO1 due to site-specific phosphorylation | 1-gen-2022 | Pacheco-Garcia, J. L.; Loginov, D.; Rizzuti, B.; Vankova, P.; Neira, J. L.; Kavan, D.; Mesa-Torres, N.; Guzzi, R.; Man, P.; Pey, A. L. | |
Interaction of letrozole and its degradation products with aromatase: chemometric assessment of kinetics and structure-based binding validation | 1-gen-2022 | De Luca, Michele; Occhiuzzi, Maria Antonietta; Rizzuti, Bruno; Ioele, Giuseppina; Ragno, Gaetano; Garofalo, Antonio; Grande, Fedora | |
The interaction of tryptophan enantiomers with model membranes is modulated by polar head type and physical state of phospholipids | 1-gen-2023 | Guglielmelli, Alexa; Bartucci, Rosa; Rizzuti, Bruno; Palermo, Giovanna; Guzzi, Rita; Strangi, Giuseppe | |
Promising Perspectives of the Antiproliferative GPER Inverse Agonist ERα17p in Breast Cancer | 1-gen-2023 | Kampa, Marilena; Lappano, Rosamaria; Grande, Fedora; Rizzuti, Bruno; Maggiolini, Marcello; Castanas, Elias; Jacquot, Yves | |
Targeting of mitochondrial fission through natural flavanones elicits anti-myeloma activity | 1-gen-2024 | Torcasio, Roberta; Gallo Cantafio, Maria Eugenia; Veneziano, Claudia; De Marco, Carmela; Ganino, Ludovica; Valentino, Ilenia; Occhiuzzi, Maria Antonietta; Perrotta, Ida Daniela; Mancuso, Teresa; Conforti, Filomena; Rizzuti, Bruno; Martino, Enrica Antonia; Gentile, Massimo; Neri, Antonino; Viglietto, Giuseppe; Grande, Fedora; Amodio, Nicola | |
Dissecting CYP1A2 Activation by Arylalkanoic Acid Prodrugs toward the Development of Anti-Inflammatory Agents | 1-gen-2024 | Occhiuzzi, Maria Antonietta; Ioele, Giuseppina; De Luca, Michele; Rizzuti, Bruno; Scordamaglia, Domenica; Lappano, Rosamaria; Maggiolini, Marcello; Garofalo, Antonio; Grande, Fedora |
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