GAROFALO, Antonio
GAROFALO, Antonio
Dipartimento di Farmacia e Scienze della Salute e della Nutrizione
A challenge in the treatment of neuropathic pain: synthesis of new photostable dihydropyridines
2020-01-01 Ioele, Giuseppina; Gözde Gündüz, Miyase; DE LUCA, Michele; Grande, Fedora; Occhiuzzi, MARIA ANTONIETTA; Garofalo, Antonio; Ragno, Gaetano
A Comparative Molecular Field Analysis Model for 6-Arylpyrrolo[2,1-d][1,5]benzothiazepines Binding Selectively to the Mitochondrial Benzodiazepine Receptor
1994-01-01 Greco, G; Novellino, E; Fiorini, I; Nacci, V; Campiani, G; Ciani, S. M.; Garofalo, Antonio; Bernasconi, P; Mennini, T.
A critical study on the application of the zero-crossing derivative spectrophotometry to the photodegradation monitoring of lacidipine
2006-01-01 Ragno, Gaetano; Ioele, Giuseppina; DE LUCA, M; Garofalo, Antonio; Grande, Fedora; Risoli, A.
A new and expeditious synthesis of 5h-pyrrolo[1,2-b][2]benzazepine derivatives
1990-01-01 Corelli, F; Garofalo, Antonio; Massa, S; Artico, M.
A pilot study on the nutraceutical properties of the Citrus hybrid Tacle® as a dietary source of polyphenols for supplementation in metabolic disorders
2019-01-01 Casacchia, Teresa; Occhiuzzi, Maria Antonietta; Grande, Fedora; Rizzuti, Bruno; Granieri, Maria Concetta; Rocca, Carmine; Gattuso, Alfonsina; Garofalo, Antonio; Angelone, Tommaso; Statti, Giancarlo
Active manganese dioxide promoted cyclization of ortho-(1H-pyrrol- 1-yl)aryl and heteroaryl carboxylic acids to 5H-pyrrolo[1,2-a][3,1] benzoxazin-5-one derivatives
2013-01-01 Grande, Fedora; Brizzi, A; Garofalo, Antonio; Aiello, Francesca
An approach to the stereo-controlled synthesis of polycyclic derivatives of L-4-thiazolidinecarboxylic acid active against HIV-1 integrase
2006-01-01 Aiello, Francesca; Brizzi, A; De Grazia, O; Garofalo, Antonio; Grande, Fedora; Sinicropi, Maria Stefania; Dayam, R; Neamati, N.
An update on small molecules targeting CXCR4 as starting points for the development of anti-cancer therapeutics.
2017-01-01 Grande, F; Giancotti, G; Ioele, G; Occhiuzzi, MARIA ANTONIETTA; Garofalo, A.
Anticancer Drugs: Recent Strategies to Improve Stability Profile, Pharmacokinetic and Pharmacodynamic Properties
2022-01-01 Ioele, Giuseppina; Chieffallo, Martina; Occhiuzzi, Maria Antonietta; De Luca, Michele; Garofalo, Antonio; Ragno, Gaetano; Grande, Fedora
Antiproliferative Action of Pyrrolobenzoxazepine derivatives in Cultured Cells: Absence of Correlation with Binding to the Peripheral-Type Benzodiazepine Binding Site
1998-01-01 Zisteres, D. M.; Hance, N; Campiani, G; Garofalo, Antonio
Benzodiazepines and Related Substances: Chemistry
2021-01-01 Grande, Fedora; Occhiuzzi, MARIA ANTONIETTA; Garofalo, Antonio.
Benzopyrroloxazines containing a bridgehead nitrogen atom as promising scaffolds for the achievement of biologically active agents
2018-01-01 Grande, Fedora; Occhiuzzi, Maria A.; Ioele, Giuseppina; Ragno, Gaetano; Garofalo, Antonio
Benzothiazine and benzothiazpine derivatives: Synthesis and preliminary biological evaluation
1993-01-01 Garofalo, Antonio; Campiani, G; Fiorini, I; Nacci, V.
Cardiovascular Characterization of Pyrrolo[2,1-d][1,5]benzothiazepine derivatives Binding Selectively to the “Peripheral-Type” Benzodiazepine Receptor (PBR). From Dual PBR Affinity and Calcium Antagonist Activity to Novel and Selective Calcium Entry Blockers
1996-01-01 Campiani, G; Fiorini, I; DE FILIPPIS, M. P.; Ciani, S. M.; Garofalo, Antonio; Nacci, V; Giorgi, G; Sega, A; Botta, M; Chiarini, A; Budriesi, R; Bruni, G; Romeo, M. R.; Manzoni, C; Mennini, T.
Cateslytin abrogates lipopolysaccharide-induced cardiomyocyte injury by reducing inflammation and oxidative stress through toll like receptor 4 interaction
2021-01-01 Rocca, Carmine; De Bartolo, Anna; Grande, Fedora; Rizzuti, Bruno; Pasqua, Teresa; Giordano, Francesca; Granieri, Maria Concetta; Occhiuzzi, Maria Antonietta; Garofalo, Antonio; Amodio, Nicola; Cerra, Maria Carmela; Schneider, Francis; Panno, Maria Luisa; Metz-Boutigue, Marie Hélène; Angelone, Tommaso
CCR5/CXCR4 dual antagonism for the improvement of HIV infection therapy
2019-01-01 Grande, Fedora; Occhiuzzi, Maria Antonietta; Rizzuti, Bruno; Ioele, Giuseppina; De Luca, Michele; Tucci, Paola; Svicher, Valentina; Aquaro, Stefano; Garofalo, Antonio
Combination effects of SC144 and cytotoxic anticancer agents
2009-01-01 Oshima, T; Cao, X; Grande, Fedora; Yamada, R; Garofalo, Antonio; Louie, S; Neamati, N.
Composition and Methods For Treating Colon and Ovarian Cancer.
2013-01-01 Neamati, N; Xu, S; Grande, Fedora; Garofalo, A.
Computational Approaches for the Discovery of GPER Targeting Compounds
2020-01-01 Grande, Fedora; Occhiuzzi, Maria A; Lappano, Rosamaria; Cirillo, Francesca; Guzzi, Rita; Garofalo, Antonio; Jacquot, Yves; Maggiolini, Marcello; Rizzuti, Bruno
Convenient synthesis of fluorazone derivatives by one-pot pyrrolation/cyclization of anthranilic acids
2011-01-01 Aiello, Francesca; Garofalo, Antonio; Grande, Fedora
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
A challenge in the treatment of neuropathic pain: synthesis of new photostable dihydropyridines | 1-gen-2020 | Ioele, Giuseppina; Gözde Gündüz, Miyase; DE LUCA, Michele; Grande, Fedora; Occhiuzzi, MARIA ANTONIETTA; Garofalo, Antonio; Ragno, Gaetano | |
A Comparative Molecular Field Analysis Model for 6-Arylpyrrolo[2,1-d][1,5]benzothiazepines Binding Selectively to the Mitochondrial Benzodiazepine Receptor | 1-gen-1994 | Greco, G; Novellino, E; Fiorini, I; Nacci, V; Campiani, G; Ciani, S. M.; Garofalo, Antonio; Bernasconi, P; Mennini, T. | |
A critical study on the application of the zero-crossing derivative spectrophotometry to the photodegradation monitoring of lacidipine | 1-gen-2006 | Ragno, Gaetano; Ioele, Giuseppina; DE LUCA, M; Garofalo, Antonio; Grande, Fedora; Risoli, A. | |
A new and expeditious synthesis of 5h-pyrrolo[1,2-b][2]benzazepine derivatives | 1-gen-1990 | Corelli, F; Garofalo, Antonio; Massa, S; Artico, M. | |
A pilot study on the nutraceutical properties of the Citrus hybrid Tacle® as a dietary source of polyphenols for supplementation in metabolic disorders | 1-gen-2019 | Casacchia, Teresa; Occhiuzzi, Maria Antonietta; Grande, Fedora; Rizzuti, Bruno; Granieri, Maria Concetta; Rocca, Carmine; Gattuso, Alfonsina; Garofalo, Antonio; Angelone, Tommaso; Statti, Giancarlo | |
Active manganese dioxide promoted cyclization of ortho-(1H-pyrrol- 1-yl)aryl and heteroaryl carboxylic acids to 5H-pyrrolo[1,2-a][3,1] benzoxazin-5-one derivatives | 1-gen-2013 | Grande, Fedora; Brizzi, A; Garofalo, Antonio; Aiello, Francesca | |
An approach to the stereo-controlled synthesis of polycyclic derivatives of L-4-thiazolidinecarboxylic acid active against HIV-1 integrase | 1-gen-2006 | Aiello, Francesca; Brizzi, A; De Grazia, O; Garofalo, Antonio; Grande, Fedora; Sinicropi, Maria Stefania; Dayam, R; Neamati, N. | |
An update on small molecules targeting CXCR4 as starting points for the development of anti-cancer therapeutics. | 1-gen-2017 | Grande, F; Giancotti, G; Ioele, G; Occhiuzzi, MARIA ANTONIETTA; Garofalo, A. | |
Anticancer Drugs: Recent Strategies to Improve Stability Profile, Pharmacokinetic and Pharmacodynamic Properties | 1-gen-2022 | Ioele, Giuseppina; Chieffallo, Martina; Occhiuzzi, Maria Antonietta; De Luca, Michele; Garofalo, Antonio; Ragno, Gaetano; Grande, Fedora | |
Antiproliferative Action of Pyrrolobenzoxazepine derivatives in Cultured Cells: Absence of Correlation with Binding to the Peripheral-Type Benzodiazepine Binding Site | 1-gen-1998 | Zisteres, D. M.; Hance, N; Campiani, G; Garofalo, Antonio | |
Benzodiazepines and Related Substances: Chemistry | 1-gen-2021 | Grande, Fedora; Occhiuzzi, MARIA ANTONIETTA; Garofalo, Antonio. | |
Benzopyrroloxazines containing a bridgehead nitrogen atom as promising scaffolds for the achievement of biologically active agents | 1-gen-2018 | Grande, Fedora; Occhiuzzi, Maria A.; Ioele, Giuseppina; Ragno, Gaetano; Garofalo, Antonio | |
Benzothiazine and benzothiazpine derivatives: Synthesis and preliminary biological evaluation | 1-gen-1993 | Garofalo, Antonio; Campiani, G; Fiorini, I; Nacci, V. | |
Cardiovascular Characterization of Pyrrolo[2,1-d][1,5]benzothiazepine derivatives Binding Selectively to the “Peripheral-Type” Benzodiazepine Receptor (PBR). From Dual PBR Affinity and Calcium Antagonist Activity to Novel and Selective Calcium Entry Blockers | 1-gen-1996 | Campiani, G; Fiorini, I; DE FILIPPIS, M. P.; Ciani, S. M.; Garofalo, Antonio; Nacci, V; Giorgi, G; Sega, A; Botta, M; Chiarini, A; Budriesi, R; Bruni, G; Romeo, M. R.; Manzoni, C; Mennini, T. | |
Cateslytin abrogates lipopolysaccharide-induced cardiomyocyte injury by reducing inflammation and oxidative stress through toll like receptor 4 interaction | 1-gen-2021 | Rocca, Carmine; De Bartolo, Anna; Grande, Fedora; Rizzuti, Bruno; Pasqua, Teresa; Giordano, Francesca; Granieri, Maria Concetta; Occhiuzzi, Maria Antonietta; Garofalo, Antonio; Amodio, Nicola; Cerra, Maria Carmela; Schneider, Francis; Panno, Maria Luisa; Metz-Boutigue, Marie Hélène; Angelone, Tommaso | |
CCR5/CXCR4 dual antagonism for the improvement of HIV infection therapy | 1-gen-2019 | Grande, Fedora; Occhiuzzi, Maria Antonietta; Rizzuti, Bruno; Ioele, Giuseppina; De Luca, Michele; Tucci, Paola; Svicher, Valentina; Aquaro, Stefano; Garofalo, Antonio | |
Combination effects of SC144 and cytotoxic anticancer agents | 1-gen-2009 | Oshima, T; Cao, X; Grande, Fedora; Yamada, R; Garofalo, Antonio; Louie, S; Neamati, N. | |
Composition and Methods For Treating Colon and Ovarian Cancer. | 1-gen-2013 | Neamati, N; Xu, S; Grande, Fedora; Garofalo, A. | |
Computational Approaches for the Discovery of GPER Targeting Compounds | 1-gen-2020 | Grande, Fedora; Occhiuzzi, Maria A; Lappano, Rosamaria; Cirillo, Francesca; Guzzi, Rita; Garofalo, Antonio; Jacquot, Yves; Maggiolini, Marcello; Rizzuti, Bruno | |
Convenient synthesis of fluorazone derivatives by one-pot pyrrolation/cyclization of anthranilic acids | 1-gen-2011 | Aiello, Francesca; Garofalo, Antonio; Grande, Fedora |