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Titolo Data di pubblicazione Autore(i) File
Progettazione e Sintesi di Nuovi Inibitori dell’Istone Deacetilasi 1-gen-2008 Aiello, Francesca; Garofalo, A; Grande, Fedora
Design and Synthesis of Pyrroloquinoxaline Based as Anticancer Agents 1-gen-2008 Aiello, Francesca; Garofalo, A.; Grande, F.
Discovery of Novel Anticancer Compounds Based on Quinoxalinhydrazide Pharmacophore 1-gen-2008 Deng, Jiexi; Taheri, L.; Grande, F.; Aiello, F; Garofalo, A.; Neamati, N.
Naphthoxazepine Inhibitors of HIV-1 Integrase: Synthesis and Biological Evaluation 1-gen-2008 Garofalo, A; Grande, Fedora; Brizzi, A; Aiello, Francesca; Dayam, R; Neamati, N.
Small molecules anti-HIV therapeutics targeting CXCR4 1-gen-2008 Grande, Fedora; Garofalo, Antonio; Neamati, N.
Design of anticancer drugs based on a chromatin-remodeling mechanism 1-gen-2009 Aiello, Francesca; Garofalo, Antonio; Grande, Fedora
Synthesis and biological evaluation of 1,3-Indandione derivatives as acetylcholinesterase inhibitors 1-gen-2009 Caruso, A; Garofalo, A; Grande, F; Anzini, M; Ortuso, F; Alcaro, S; Panno, Antonella; Saturnino, C; Sinicropi, M. S.
Design, Synthesis and Biological Evaluation of Novel Anticancer Agents Based on APE1 Pharmacophore Model 1-gen-2009 Aiello, Francesca; Grande, Fedora; Garofalo, A.
Discovery of a Novel Quinoxalinhydrazide with Broad Spectrum of Anticancer Activity 1-gen-2009 Plasencia, C; Grande, Fedora; Oshima, T; Cao, X; Yamada, R; Sanchez, T; Aiello, Francesca; Garofalo, A; Neamati, N.
Synthesis and biological evaluation of novel hydrazide based cytotoxic agents 1-gen-2009 Grande, Fedora; Yamada, R; Cao, Xf; Aiello, Francesca; Garofalo, Antonio; Neamati, N.
Combination effects of SC144 and cytotoxic anticancer agents 1-gen-2009 Oshima, T; Cao, X; Grande, Fedora; Yamada, R; Garofalo, Antonio; Louie, S; Neamati, N.
Efficient synthesis of 9H-pyrrolo[1,2-a]indol-9-one derivatives based on active manganese dioxide promoted intramolecular cyclization 1-gen-2010 Aiello, Francesca; Garofalo, Antonio; Grande, Fedora
Direct cyclization of ortho-(1H-pyrrol-1-yl)aryl and heteroaryl carboxylic acids into fused pyrrolizinones 1-gen-2010 Aiello, Francesca; Garofalo, A; Grande, Fedora
SC144: The first orally active small molecule gp130 inhibitor for the treatment of ovarian cancer. 1-gen-2011 Xu, S; Grande, Fedora; Garofalo, A; Neamati, N.
Esteri di acidi grassi insaturi e ormoni androgeni potenzialmente utili nel trattamento del dolore 1-gen-2011 Aiello, Francesca; Aloisi, A. M.; Anzini, M; Garofalo, A; Grande, Fedora; Petroni, A.
One-pot transformation of anthranilic acids to fluorazone derivatives, valuable intermediates for the synthesis of anticancer agents. 1-gen-2011 Aiello, Francesca; Garofalo, A; Grande, Fedora
Convenient synthesis of fluorazone derivatives by one-pot pyrrolation/cyclization of anthranilic acids 1-gen-2011 Aiello, Francesca; Garofalo, Antonio; Grande, Fedora
Small-Molecule Inhibitors of p53-MDM2 Interaction: the 2006-2010 Update 1-gen-2011 Millard, M; Pathania, D; Grande, Fedora; Xu, S; Neamati, N.
Mechanistic characterization of SC144 in colon cancer 1-gen-2012 Xu, S; Oshima, T; Grande, F; Neamati, N; Garofalo, Antonio
Valutazione della tossicità acuta di piante medicinali mediante microtox test. 1-gen-2012 Ioele, Giuseppina; DE LUCA, M; Grande, Fedora; Ragno, Gaetano
Mostrati risultati da 21 a 40 di 163
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