Sfoglia per Autore
Progettazione e Sintesi di Nuovi Inibitori dell’Istone Deacetilasi
2008-01-01 Aiello, Francesca; Garofalo, A; Grande, Fedora
Design and Synthesis of Pyrroloquinoxaline Based as Anticancer Agents
2008-01-01 Aiello, Francesca; Garofalo, A.; Grande, F.
Discovery of Novel Anticancer Compounds Based on Quinoxalinhydrazide Pharmacophore
2008-01-01 Deng, Jiexi; Taheri, L.; Grande, F.; Aiello, F; Garofalo, A.; Neamati, N.
Naphthoxazepine Inhibitors of HIV-1 Integrase: Synthesis and Biological Evaluation
2008-01-01 Garofalo, A; Grande, Fedora; Brizzi, A; Aiello, Francesca; Dayam, R; Neamati, N.
Small molecules anti-HIV therapeutics targeting CXCR4
2008-01-01 Grande, Fedora; Garofalo, Antonio; Neamati, N.
Design of anticancer drugs based on a chromatin-remodeling mechanism
2009-01-01 Aiello, Francesca; Garofalo, Antonio; Grande, Fedora
Synthesis and biological evaluation of 1,3-Indandione derivatives as acetylcholinesterase inhibitors
2009-01-01 Caruso, A; Garofalo, A; Grande, F; Anzini, M; Ortuso, F; Alcaro, S; Panno, Antonella; Saturnino, C; Sinicropi, M. S.
Design, Synthesis and Biological Evaluation of Novel Anticancer Agents Based on APE1 Pharmacophore Model
2009-01-01 Aiello, Francesca; Grande, Fedora; Garofalo, A.
Discovery of a Novel Quinoxalinhydrazide with Broad Spectrum of Anticancer Activity
2009-01-01 Plasencia, C; Grande, Fedora; Oshima, T; Cao, X; Yamada, R; Sanchez, T; Aiello, Francesca; Garofalo, A; Neamati, N.
Synthesis and biological evaluation of novel hydrazide based cytotoxic agents
2009-01-01 Grande, Fedora; Yamada, R; Cao, Xf; Aiello, Francesca; Garofalo, Antonio; Neamati, N.
Combination effects of SC144 and cytotoxic anticancer agents
2009-01-01 Oshima, T; Cao, X; Grande, Fedora; Yamada, R; Garofalo, Antonio; Louie, S; Neamati, N.
Efficient synthesis of 9H-pyrrolo[1,2-a]indol-9-one derivatives based on active manganese dioxide promoted intramolecular cyclization
2010-01-01 Aiello, Francesca; Garofalo, Antonio; Grande, Fedora
Direct cyclization of ortho-(1H-pyrrol-1-yl)aryl and heteroaryl carboxylic acids into fused pyrrolizinones
2010-01-01 Aiello, Francesca; Garofalo, A; Grande, Fedora
SC144: The first orally active small molecule gp130 inhibitor for the treatment of ovarian cancer.
2011-01-01 Xu, S; Grande, Fedora; Garofalo, A; Neamati, N.
Esteri di acidi grassi insaturi e ormoni androgeni potenzialmente utili nel trattamento del dolore
2011-01-01 Aiello, Francesca; Aloisi, A. M.; Anzini, M; Garofalo, A; Grande, Fedora; Petroni, A.
One-pot transformation of anthranilic acids to fluorazone derivatives, valuable intermediates for the synthesis of anticancer agents.
2011-01-01 Aiello, Francesca; Garofalo, A; Grande, Fedora
Convenient synthesis of fluorazone derivatives by one-pot pyrrolation/cyclization of anthranilic acids
2011-01-01 Aiello, Francesca; Garofalo, Antonio; Grande, Fedora
Small-Molecule Inhibitors of p53-MDM2 Interaction: the 2006-2010 Update
2011-01-01 Millard, M; Pathania, D; Grande, Fedora; Xu, S; Neamati, N.
Mechanistic characterization of SC144 in colon cancer
2012-01-01 Xu, S; Oshima, T; Grande, F; Neamati, N; Garofalo, Antonio
Valutazione della tossicità acuta di piante medicinali mediante microtox test.
2012-01-01 Ioele, Giuseppina; DE LUCA, M; Grande, Fedora; Ragno, Gaetano
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